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اثرات ضد دردی گاباپنتین و
ایبوپروفن بر درد بعد از درمان ریشه
در سال ۲۰۰۲ به پزشکان اجازه داده شد که از این دارو
برای کاهش درد ناشی از ابتلا به زونا (نورالژی هرپسی)
استفاده کنند. کمتراز 100 میلی
گرم تقریباً 7/1 ساعت است ، در حالی که Tmax در دوزهای
بالاتر3 تا 4 ساعت است. غذا به میزان
قابل توجهی بر Tmax گاباپنتین تأثیر نمی گذارد.
گاباپنتین ممکن است باعث شود احساس خواب آلودگی و کسالت
داشته باشید و قدرت تصمیم گیری تان تحت تأثیر
قرار بگیرد.
برای درمان حتماً لازم است که به پزشک مراجعه کنید و از خود درمانی بپرهیزید.
متابولیسم گاباپنتین متابولیسم کمی دارد یا اصلاً متابولیسم نمی شود.
برعکس ، گاباپنتین اناکاربیل ، که به عنوان پیش داروی گاباپنتین عمل می کند ، برای فعال شدن
باید تحت هیدرولیز آنزیمی قرار
گیرد.این کار از طریق استرازهای غیر اختصاصی در روده و به میزان کمتری در کبد انجام می شود.
گاباپنتین برای اولین بار در
سال 1993 مورد استفاده قرار گرفت. این دارو از سال 2004 به
عنوان دارو در ایالات متحده در دسترس است.
در سال 2017 ، با بیش از 46 میلیون نسخه ، یازدهمین داروی معمولاً تجویز شده در ایالات متحده بود.
هدف این مطالعه مقایسه تأثیر گاباپنتین و پرگابالین بهعنوان پیشدارو
در پیشگیری از پاسخهای همودینامیک ناشی از لارنگوسکوپی و لولهگذاری بود.
مرالژيا پارسنتيكا ( درد يا تحريك پذيرى در ران پا ) ، قطع عضو ، و سر درد
، نيز مفيد واقع مى شود . طبق گزارش ها ، اين دارو در درمان بعضى موارد
پروريتوس ( خارش ) مزمن مفيد واقع
شده است . ما فقط شواهدی را با کیفیت بسیار
پائین در اختیار داریم و درباره تخمین سودمندی و آسیب ناشی از دارو
به علت دادههای ناکافی، بسیار نامطمئن هستیم.
شواهد ناکافی وجود دارد که بتواند از توصیه گاباپنتین
به افراد مبتلا به فیبرومیالژیا برای کاهش درد حمایت
کند. 4- این دارو ممکن است روی نتیجه آزمایش پروتئین ادرار اثر بگذارد.
سلام دکتر.مدتی است که به خاطر دیسک
کمر گاباپنتین ۱۰۰مصرف میکنم بعضی شبها احساس تنگی نفس میکنم انگار کسی داره خفه ام میکنه به
نظر شما مال مصرف این قرص است. قبل از مصرف گاباپنتین ، حتماً در
مورد تمام نسخه های دارویی ، بدون نسخه و سایر
داروهای مصرف شده به پزشک و داروساز
خود بگویید. همچنین در مورد هر نوع ویتامین ، گیاهان و مکمل های استفاده شده به آنها بگویید.
به اشتراک گذاشتن این اطلاعات می تواند در جلوگیری
از تعامل بالقوه به شما کمک کند.
اگر در مورد تداخلات دارویی که ممکن است روی شما تأثیر بگذارد سؤال دارید ،
از پزشک یا داروساز خود بپرسید.
این مطالعه شواهد خوبی از
توصیه به مصرف گاباپنتین روزانه با دوزهای
1200 تا 2400 میلیگرم برای کاهش درد در افراد مبتلا به فیبرومیالژیا که
حمایت یا آن را رد کند، ارائه نکرد.
بنابراین دردی ایجاد میشود که
نه تنها راه رفتن را مختل میکند بلکه میتواند کاملاً شدید باشد.
قطع ناگهانی آن ممکن است باعث بازگشت علائم
بیمار شود. این دارو ممکن است روی نتیجه آزمایش پروتئین ادرار اثر بگذارد.
کودکان و سالخوردگان به عوارض جانبی ناشی از این دارو حساس تر هستند.
این دارو به عنوان ضد درد معمولی
یا در درد ناشی از بیماریی آرتریت
کاربرد ندارد. 2-گاباپنتن را می توانید همراه غذا یا بدون آن میل کنید.
در ادامه به برخی از سوالات
درباره گاباپنتین پاسخ دادهشدهاست.
با ما همراه باشید و به دانش خود درباره
داروی گاباپنتین بیفزایید.
تعداد زیادی از افرادی که به کمپهای ترک اعتیاد مراجعه میکنند، به خاطر سوء مصرف گاباپنتین است.
این دارو در دوران بارداری فقط در صورت صلاحدید و تجویز پزشک باید مصرف شود.
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